Noj qab haus huv, Npaj
Cov tshuaj "Ofloxacin": tus neeg mob testimonials. Cov lus qhia rau kev siv ntawm cov tshuaj tua kab mob "Ofloxacin"
Kev npaj "Ofloxacin" kev cov neeg mob uas feem ntau zoo, nruab nrab yog cov antimicrobial neeg sawv cev los ntawm cov pab pawg neeg ntawm fluoroquinolones sab spectrum ntawm kev ua si. Cov tshuaj muaj feem xyuam rau cov DNA gyrase - kab mob fragment, muab supercoiling thiab yog li ntawd lub stability ntawm cov kab mob DNA (raws li ib tug tshwm sim ntawm destabilization ntawm cov DNA strand tuag).
pharmacodynamics
Txhais tau hais tias "Ofloxacin" - ib tug tshuaj tua kab mob zoo nrog rau kev hwm mus kab mob uas tsim beta-lactamase, raws li zoo raws li ceev ceev-loj hlob atypical mycobacteria. Yuav kom cov tshuaj yog rhiab, feem ntau Gram-tsis zoo kab mob, xws li kab mob uas yog resistant rau methicillin thiab lwm yam tshuaj tua kab mob. Streptococci, Enterococci, thiab Mycobacterium tuberculosis yog yus muaj los ntawm tsis ruaj tsis khov nyhav mus rau yeeb tshuaj "Ofloxacin". Xyuas ntawm cov kws kho mob qhia tias nyob rau hauv cov kev kho mob ntawm co kab mob tshwm sim los ntawm peptostreptokokki, peptokokki thiab lwm yam anaerobes, cov tshuaj no feem ntau yog tsis zoo.
tshuaj
Thaum tau txais cov medicament mus rau hauv lub haum yog tiav (95 feem pua) thiab ceev ceev. Bioavailability - ntau tshaj 96 feem pua. Kev sib raug zoo rau ntshav cov nqaijrog - 25 feem pua. Tom qab ib mus rau ob teev tom qab qhov ncauj thawj coj ntawm lub siab tshaj plaws concentration attained. Nws yog KOOB-dependent: ib siv ob puas, plaub los yog rau pua milligrams ntawm cov tshuaj concentration twb feem 2.5, 5 los yog 6.9 ug / ml.
Khoom noj khoom haus noj yuav cuam tshuam rau haum ntawm lub sab ntawm ib tug slowdown, tab sis tsis muaj teeb meem loj ntxim rau cov bioavailability. Kev npaj "Ofloxacin" - ib tug tshuaj tua kab mob muaj ib tug txiav txim volume ntawm tis (ib puas gallons), yog li ntawd lub xeem yog kev npaj yuav luag tag nrho cov nqi penetrates dawb do rau hauv lub hlwb. Qhov siab tshaj plaws ntau yog nyob rau hauv cov ntaub so ntswg, lub cev thiab nruab nrog cev: nyob rau hauv lub hlwb (alveolar macrophages, leukocytes), tej nqaij mos, daim tawv nqaij, pob txha, ua pa system, pelvic thiab mob plab kab noj hniav, cov qaub ncaug, prostatic kua, zis, kua tsib. Lub medicament zoo penetrates rau hauv lub placental thiab cov ntshav-hlwb barrier, yog secreted los ntawm ob lub mis mis nyuj, thiab hlwb txha nqaj qaum kua nkag mus rau ntawm qhov uas tsis yog-kub lug thiab kub lug hlwb week (14 mus rau 60 feem pua).
Hais txog 5 feem pua ntawm cov tshuaj no yog metabolized nyob rau hauv lub siab mus rau daim ntawv dimetilofloksatsina thiab N-oxide ntawm ofloxacin. Tsis hais txog ntawm cov tshuaj ib nrab-lub neej yog ntawm plaub thiab ib tug ib nrab mus rau xya teev. Tso zis unchanged tshuaj nyob rau hauv ib tug npaum li ntawm 75-90 feem pua ntawm ob lub raum, nyob rau hauv ib tug npaum li ntawm 4 feem pua - nyob rau hauv lub bile. Tsawg tshaj li 20 feem pua ntawm cov extrarenal clearance. Tom qab ib tug tib koob tshuaj ntawm ob puas milligrams ntawm tus neeg saib xyuas yog detectable nyob rau hauv cov zis rau 20-24 teev. Nyob rau hauv cov ntaub ntawv ntawm hepatic los yog lub raum feem tej zaum yuav tub ceevxwm. Thaum lim ntshav yog muab tshem tawm los ntawm 10 mus rau 30 feem pua ntawm cov tshuaj.
indications rau
Nyob rau hauv kab thiab inflammatory kab mob tshwm sim los ntawm ntau yam kab mob, qhia ntawv thov medicament "Ofloxacin". Xyuas tau qhia hais tias nws yog zoo heev rau ua pa ib ntsuj av tau kab mob (mob ntsws, ntsws), Upper pa ib ntsuj av tau (otitis media, sinusitis, laryngitis, pharyngitis). Muab tshuaj nyob rau hauv tej nqaij mos txhab, pob qij txha, pob txha, daim tawv nqaij, biliary ib ntsuj av tau, mob txeeb zig (urethritis, cystitis), mob raum (pyelonephritis), mob plab kab noj hniav, genitalia (orchitis, colpitis, epididymitis), hu ua pelvic kabmob (salpingitis, prostatitis, cervicitis, endometritis, oophoritis, tsis).
Tsis tas li ntawd zoo tshuaj rau ureaplasmosis, chlamydia, gonorrhea. Siv nws rau kev tiv thaiv ntawm tus kab mob nyob rau hauv cov neeg mob uas mob ntawm lub cev raws li txoj cai (xws li cov neutropenia).
Cov tshuaj daim ntawv. qauv
Tus tso tawm ntawm medicament yog nyob rau hauv daim ntawv ntawm cov loj dawb los yog yuav luag dawb zaj duab xis-coated ntsiav tshuaj biconvex hloov puab. Tus ntoo khaub lig sectional hnov ob khaubncaws sab nraud povtseg, yog ib tus uas muaj ib tug yellowish tint. Active tivthaiv ua raws li ofloxacin. Ib tug ntsiav tshuaj muaj nyob rau hauv cov huab hwm coj ntawm 200 los yog 400 mg. Me khoom xyaw yog primelloza (croscarmellose sodium), microcrystalline cellulose, Aerosil (colloidal silicon dioxide), silica titania, povidone, hydroxypropyl methylcellulose (hypromellose), talc, magnesium stearate, polyethylene glycol 4000 (macrogol). Ib tug poj kom zoo dua ntawm cov tshuaj "Ofloxacin" - nqi. Ntsiav tshuaj muaj 200 mg ntawm active tshuaj yog ib tug nruab nrab ntawm 16-20 rubles ib 10 daim, thiab cov neeg uas muaj 400 milligrams ofloxacin, yuav raug nqi txog 50-55 rubles ib 10 daim.
"Ofloxacin" tshuaj. Cov lus qhia rau kev siv
Ntsiav tshuaj yuav tsum haus dej haus ua ntej los yog tom qab ib tug noj mov. Lawv yuav tsum tau nqos tag nrho, tsis muaj zom, thiab haus dej nyob rau hauv me me qhov ntau. Cov tshuaj yuav tsum tau xaiv ib lub zuj zus nyob rau hauv lub heev ntawm tus kab mob, lub chaw ntawm tus kab mob, tus neeg mob lub kev mob, lub raum muaj nuj nqi, daim siab, thiab kab mob rhiab heev.
Raws li ib tug txoj cai, cov kev kho mob ntawm "ofloxacin" yog ua rau xya mus rau kaum hnub. Tus neeg laus hnub kho kom tsawg ntawm ob puas, rau puas milligrams ob zaug ib hnub twg. Cov koob tshuaj tej zaum yuav muab tau ntau zog mus rau yim milligrams nyob rau hauv cov ntaub ntawv ntawm ib tug kab mob, los yog hais tias tus neeg mob yog tus neeg rog. A koob tshuaj plaub milligrams yuav npaum li cas nyob rau ib zaug, dua li nyob rau hauv thaum sawv ntxov.
Cov neeg mob uas raum tsis ua haujlwm ib zaug tsis tau ntau tshaj li ob puas milligrams ntawm cov tshuaj, lub siab tshaj plaws tshuaj txhua txhua hnub nyob rau hauv hepatic puas - plaub puas milligrams. Tom qab lub disappearance ntawm cov tsos mob thiab normalization ntawm kub, txawm rau ob los yog peb hnub yuav tsum kho.
Sab los. Testimonials
Tsis yog txhua txhua tus neeg mob cov tshuaj "Ofloxacin" zoo taus. Xyuas ntawm ib co neeg muaj cov ntaub ntawv uas cov tshuaj ua rau mob taub hau, xeev siab, ntuav, raws plab, tshee, xws li loog loog ntawm extremities. Nyob rau hauv ib feem ntawm lub digestive system yuav tsim raws li mob plab, gastralgia, tsam plab, cholestatic daj ntseg, anorexia, hyperbilirubinemia, pseudomembranous enterocolitis, thiab lub paj hlwb - tsis muaj zog, tu-sauv, mob siab heev npau suav, psychotic tshua, ntxhov siab, ntxhov siab vim, tsis meej pem, phobias, hallucinations, kev nyuaj siab.
Nyob rau hauv tas li ntawd, muaj yog kev pheej hmoo ntawm kev ua txhaum ntawm lub cev muaj zog system (arthralgia, tendonitis, myalgias), tsis totaub (saj mob, pom xim, lub rooj sib hais, tshuav nyiaj li cas, tsis hnov tsw), vascular system thiab lub plawv (yuav txo tau nyob rau hauv cov ntshav siab, tachycardia), daim tawv nqaij (dermatitis, taw tes hemorrhage, papular pob liab liab), ntawm hematopoiesis (thrombocytopenia, anemia, leukopenia). Tom qab tau txais "Ofloxacin" tshuaj (xyuas paub meej tias qhov no), nyob rau hauv tej zaum nws zoo nkaus li khaus khaus tawv nqaij, bronchospasm, urticaria.
Contraindications
Tau txais medicament txwv tsis pub intolerance ofloxacin thiab lwm yam fluoroquinolone derivatives, nyob rau hauv cov ntaub ntawv ntawm tsis muaj peev xwm ntawm glucose-6-phosphate dehydrogenase, qaug dab peg, txhab ntawm lub tendons, txo qaug dab peg chaw pib. Nyob rau hauv tas li ntawd, koj yuav tsis tau cov tshuaj "Ofloxacin" cev xeeb tub thiab lactating cov poj niam, cov me nyuam nyob rau hauv lub hnub nyoog ntawm kaum yim. Nrog ceev faj npaj tshuaj rau lub plawv mob nyob rau hauv lub hlwb, cerebral vascular atherosclerosis, raum tsis ua hauj lwm nyob rau hauv mob Cns txhab organic xwm.
Medicament "Ofloxacin" nyob rau hauv ib tug ureaplasma. Xyuas
Qhov loj tshaj plaws yog tias cov neeg hais tias, siv ib yam khoom - nws yog nws ceev nyhuv. Cov neeg mob qhia tias qhov kawg yog hnov twb nyob rau hauv peb los yog plaub hnub. Tab sis nws yog tsim nyog los ceeb toom hais tias qhov no tsis tau txhais hais tias qhov pib ntawm kev kho. Cov neeg mob uas tau tso tseg tsis haus cov ntsiav tshuaj, tsis tas yuav mus los ntawm tag nrho cov hoob kawm, ces dua tej ureaplasmosis cov tsos mob, vim hais tias cov kab mob tsis tau kiag li tshem tawm.
ceev faj
Thaum mob ntsws provoked los ntawm pneumococcus, cov tshuaj tsis zoo. Tsis tas li ntawd, nws tsis yog qhia rau cov kev kho mob ntawm mob tonsillitis. Nws yog tsim nyog mus lawm tshuaj no yog tias nyob rau hauv lub keeb kwm yav dhau ntawm nws mus kawm ua ib tug tsis haum cov tshuaj tiv thaiv, tus Cns teeb meem, pseudomembranous mob plab. Cov poj niam thov txhais tau tias "Ofloxacin", nws yog tsis pom zoo kom siv tampons, vim hais tias nyob rau hauv cov ntaub ntawv no muaj ib tug raug mob ntawm cov qhov ncauj tawm.
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