Noj qab haus huv, Npaj
"Thiotriazoline": cov lus qhia rau kev siv
Koj kos npe rau cov tshuaj "Thiotriazoline"? nyob rau kev siv ntawm cov tshuaj no daim ntawv qhia yuav tsum tau piav nyob rau hauv kom meej nyob rau hauv lub tam sim no tsab xov xwm. Nyob rau hauv tas li ntawd, peb yuav qhia rau koj txog cov ntawv no nyob rau hauv uas cov tshuaj nkag mus rau hauv hais tias muag, uas nws muaj indications, tshwm sim thiab contraindications.
Muaj pes tsawg leeg ntawm cov tshuaj ntim thiab tso tawm daim ntawv
Nyob rau hauv dab tsi daim ntawv tso tawm medicament "Thiotriazoline"? Cov lus qhia qhia hais tias nws muaj ib tug xov tooj ntawm ntau yam ntaub ntawv. Cov feem nrov yog:
- Ib tug tov npaj rau intramuscular thiab tso dej txhaj tshuaj. 1 ml ntawm tus neeg saib xyuas muaj 0,025 g Thiotriazoline. Tsis tas li ntawd ib tug medicament thiab yeem Cheebtsam nyob rau hauv daim ntawv ntawm cov dej rau txhaj tshuaj. Cov tshuaj no muaj nyob rau 4 ml ampoules (muab tso rau hauv lub thawv).
- "Thiotriazoline" qhov muag dauv. Los ntawm kev siv ntawm xws li ib tug qhia txhais tau tias hais tias 5 ml muaj 50 mg ntawm yeeb tshuaj Thiotriazoline, raws li zoo li lwm yam tshuaj. Cov tshuaj no yog muag nyob rau hauv yas hwj, droppers, muab tso rau hauv ib lub cardboard lub thawv.
- "Thiotriazoline" tshuaj. Cov lus qhia rau daim ntawv no ntawm cov tshuaj hais tias nyob rau hauv ib tug dawb yeej ntsiav tshuaj nrog ib tug ca saum npoo uas muaj 100 mg morfoliniymetiltriazoliltioatsetata, los yog thiaj li hu ua Thiotriazoline. Raws li ntxiv Cheebtsam ntawm lub medicament ua qos starch, microcrystalline cellulose, tsis tshua muaj molecular yuag povidone, calcium stearate thiab sucrose. Raws li ib tug txoj cai, nyob rau hauv ib tug duab los qhia pob muaj 50 ntsiav tshuaj.
pharmacodynamics
Yuav ua li cas yog lub tshuaj raws li "Thiotriazoline"? Cov lus qhia rau Siv hais tias qhov no antioxidant tshuaj. Nws high efficiency yog vim cov antioxidant, antiischemic, immunomodulatory thiab daim nyias nyias stabilizing zog.
Saib cov tshuaj tiv thaiv kev puas tsuaj ntawm hepatocytes, muaj txhawb rau lawv rov qab, thiaj li muaj cov degree ntawm fatty infiltration, uas ua rau normalization ntawm cov protein, carbohydrate, lipid thiab xim pauv, thiab thiaj li yuav ua rau muaj tus kab necrosis tsentrolobulyarnyh ib lub cev xws li hauv lub siab. Tsis tas li ntawd, active tshuaj pab txoj kev rho tawm thiab synthesis ntawm cov kua tsib, normalizes nws muaj pes tsawg leeg (tshuaj).
Lub zog ntawm cov tshuaj
Yuav ua li cas muaj lub zog ntawm cov tshuaj "Thiotriazoline"? Cov lus qhia rau kev siv ntawm cov tshuaj yuav tsum tau rau kev nyeem ntawv. Tom qab tag nrho, tsuas yog los ntawm nws koj muaj peev xwm kawm txog dab tsi qhov suav hais tias cov tshuaj txo inhibition ntawm oxidative dab nyob rau hauv lub Krebs voj voog, ua kom cov intracellular ATP nyiaj, raws li zoo raws li tej qhov ua kom (nyiaj) glycolysis co.
Tsis tas li ntawd nco ntsoov tias tom qab noj cov tshuaj active tshuaj pib qhib lub antioxidant system, Sibhawm inhibit oxidative dab nyob rau hauv lub ischemic chaw ntawm lub cev. Nyob rau hauv tas li ntawd, cov tshuaj no pab txoj kev cov khoom (rheology) ntawm cov ntshav vim qhib rua ntawm lub fibrinolytic system.
Cov antioxidant zog ntawm cov tshuaj manifested los ntawm qhov tseeb hais tias cov qauv ntawm cov molecule yog tiotrazolina leej faj ions, tsiag ntawv los ntawm oxidation thiab txo nta, raws li zoo raws li tertiary nitrogen, uas binds ib tug ntau npaum li cas ntawm hydrogen ions.
Peb kuj yuav tsum nco ntsoov tias lub active tshuaj tivthaiv yuav hnov mob nrog lipid radicals thiab reactive pa hom. Qhov no yog vim ib tug qhia tau txo thaj chaw ntawm lub thiol pab pawg neeg. Nyob rau hauv tas li ntawd, lub medicament tiv thaiv lub tsim ntawm reactive pa hom, xws antiradical reactivating enzymes li catalase, glutathione peroxidase thiab superoxide dismutase.
tshuaj
Seb tshuaj yog absorbed "Thiotriazoline"? Instruction hais tias lub sij hawm poluabsorbtsii tshuaj yog 30 feeb thiab bioavailability - 65,5%.
Maximum ntshav concentration txhais tau tias yog tiav los ntawm 1.4 lub sij hawm tom qab thawj coj. Kev sib txuas lus nrog cov nqaijrog tsis pub tshaj 10%.
Nyob rau hauv loj qhov ntau, cov tshuaj accumulates nyob rau hauv cov ntaub so ntswg ntawm daim siab, lub plawv, cov nyuv, tus po thiab ob lub raum, thiab me me - nyob rau hauv cov hnyuv thiab cov ntsws. Thiotriazoline tas tsuas yog los ntawm ob lub raum.
zaj lus tim khawv
Yog hais tias muaj yog hloov yuav raug muab tso tshuaj, tshuaj thiab qhov muag dauv "Thiotriazoline"? nyob rau kev siv ntawm cov ntaub ntawv ntawm kev qhia ntawv qhia tau hais tias cov nram qab no indications:
- mob npuas paug;
- tshuaj lom lub siab puas, dej, kis, thiab tshuaj (e.g., tom qab tau txais tshuaj tua kab mob, antiviral tshuaj, anti-TB thiab anti-mob cov neeg ua hauj, qhov ncauj contraceptives thiab tricyclic antidepressants);
- mob kis tus kab mob siab;
- alcoholic kab mob siab mob hauj sim mus rau tsawg heev kev ua si;
- fatty siab degeneration.
Indications rau kev siv tshuaj:
- corneal kab mob;
- kub nyhiab los yog qhov muag raug mob;
- kab conjunctivitis.
Yog vim li cas tseem siv ophthalmic tshuaj "Thiotriazoline"? Cov lus qhia (rau yuav yuav tau nyob tej lub tsev muag tshuaj) qhia hais tias qhov no tshuaj yog feem ntau kws kho rau cov kev tiv thaiv ntawm qhuav qhov muag, eyestrain, thiab lwm yam inflammatory kab mob ntawm nrig txog kev pom cov kabmob.
Cov tshuaj ntsiav tshuaj
Yuav ua li cas kuv yuav tsum tau siv "Thiotriazoline" ntsiav tshuaj? Phau ntawv muaj cov lus qhia tias cov tshuaj yuav tsum tau noj xwb hauv. Raws li ib tug txoj cai, thiotriazolin taw 1 los yog 2 ntsiav tshuaj plaub zaug ib hnub twg rau 25-30 hnub.
Lub caij ntawm kev kho mob nrog rau qhov no neeg sawv cev yuav tsum tau txiav txim los ntawm ib tug kws kho mob rau ib tug neeg hauv paus (nyob ntawm seb lub kawm thiab heev ntawm uas twb muaj lawm tus kab mob).
Cov tshuaj tov "Thiotriazoline": cov lus qhia rau kev siv
Tshuaj "Thiotriazoline" ua intramuscularly los yog intravenously. Lawv ntau npaum txiav txim los ntawm tus kws kho mob (nyob ntawm seb tus kab mob). Heart attack myocardial infarction thiab kab mob siab tshuaj maj mam txhaj intravenously nyob rau hauv 2 ml 2-3 zaug ib hnub twg. Nyob rau hauv mob npuas paug medicament yog muab intramuscularly (2 ml 2-3 zaug ib hnub twg). Hoob no ntawm kev kho mob yog 60 hnub.
Qhov muag rau "Thiotriazoline": cov lus qhia rau kev siv
Qhov muag rau "Thiotriazoline" instilled rau hauv lub conjunctival sac. Feem ntau, cov tshuaj rau cov neeg laus yog 2 ncos txog li 4 lub sij hawm ib hnub twg. Nrog kev xav txog cov me nyuam, cov nyiaj ntawm cov tshuaj yog txiav txim los ntawm ib tug cov menyuam yaus. Lub caij ntawm kev kho mob nrog lub qhov muag dauv thiab yuav tsum muab ntsia los ntawm cov kws kho mob.
Raws li ib tug txoj cai, lub caij ntawm kev kho mob nrog rau qhov no uas yog tsis muaj ntau tshaj li 2 lub lis piam. Tab sis, yog hais tias tsis muaj txoj kev txhim kho yog cai, hauv chav kawm yuav raug ncua txog li ib hlis.
Nyob rau hauv rooj plaub uas nws kim heev txhab nrig txog kev pom nruab nrog cev thiab loj heev, ces dropwise Ntxiv rau ocular tshuaj muab (lwm npaj).
Rau kev tiv thaiv ntawm qhuav ntawm lub qhov muag week (thaum ua hauj lwm ntawm ib lub computer), koj yuav tsum tau siv ib yam tshuaj 2 ncos thaum lub sij hawm lub hnub nrog ib tug caij nyoog ntawm 2 teev.
phiv
Yuav ua li cas yog cov kev phiv los ntawm cov tshuaj yuav ua rau "Thiotriazoline" (tshuaj)? Cov lus qhia rau cov qauv no yuav qhia tau tias cov tshuaj yog zoo taus nrog hwm. Txawm li cas los, siv qhov suav hais tias cov tshuaj yuav tseem tshwm sim undesired tshua.
- Central tshee system: kiv kiv taub hau, tsis muaj zog, ringing nyob rau hauv lub pob ntseg.
- Hnyuv: qhov ncauj qhuav, xeev siab, tsam plab.
- Hlab ntsha thiab lub plawv, muaj ntshav siab, tachycardia, arrhythmia, lub plawv mob.
- Ua pa system: mob hawb pob thiab ua tsis taus pa.
- Kev tsis haum tshuaj: kub taub hau, npau taws me ntsis kev tshua, angioedema.
- Local tshua: liab thiab tingling nov ntawm nqaij tawv ntawm lub qhov koob.
- Dermatological tshua: daim tawv nqaij yaug kais dej, khaus, ua xua.
Raws li rau qhov muag dauv, uas nyob rau lawv ib feem rau sab los muaj cai.
tshuaj cov kev sib tshuam
Raws li kws txawj, cov tshuaj "Thiotriazoline" yuav siv tau nyob rau hauv nrog yooj yim tshuaj npaj rau cov kev kho mob ntawm coronary mob plawv. Qhov no yog vim lub fact tias hais tias cov tshuaj yog ib tug cardioprotective neeg sawv cev.
Nws yuav tsum tau muab sau tseg tias cov tshuaj yog tso cai rau yuav siv ib txhij nrog rau cov tshuaj uas muab rau cov uas tsim nyog kev kho mob ntawm tus kab mob siab etiology.
Qhov muag rau "Thiotriazoline" yuav raug muab tso rau cev xeeb tub cov poj niam thiab lub sij hawm lactation. Nws yuav tsum raug hais tias tus duab ntawm lub hais tias cov khoom muaj cai siv nyob rau hauv ua ke nrog lwm yam kev kho mob txhais tau tias.
Haus dej cawv thiab tshuaj "Tiatriazolin" txhawb lwm tus txoj kev txiav txim. Nyob rau hauv no hais txog, lawv cov concomitant siv yog txwv tsis pub.
ceev faj
Muaj pes tsawg leeg muaj xws li sucrose xam tau tias yog ntsiav tshuaj (nyob rau hauv ib tug npaum li ntawm 2.8 mg ib ntsiav tshuaj). Yog li, rau cov nyiaj pab ntau tshaj txhua hnub koob tshuaj noj tshuaj yuav muaj txog 22,4 mg ntawm lub substance. Qhov tseeb yuav tsum paub cov neeg mob, cov neeg mob uas mob ntshav qab zib mellitus.
Cov kev thiab lub sij hawm ntawm cia
Kiag li tag nrho cov ntaub ntawv "Tiatriazolin" tshuaj yuav tsum muaj kev tiv thaiv los ntawm lub teeb thiab ncav cuag ntawm cov me nyuam ntawm ib tug kub ntawm los ntawm 14 mus rau 26 degrees. Lub txee lub neej ntawm cov tshuaj yog 3 lub xyoo.
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