Noj qab haus huv, Npaj
Hauj lwm thiab cov lus qhia rau kev siv: "Albarel"
Yuav ua li cas yog cov tshuaj "Albarel"? Cov lus qhia rau kev siv thiab piav qhia txog cov tshuaj yuav tsum tau muab los sib tham li hauv qab no. Peb kuj qhia koj txog cov ntawv no nyob rau hauv uas cov tshuaj yog tso tawm dua nws yog zoo tshaj plaws yuav ua li cas cov neeg mob teb rau nws.
Muaj pes tsawg leeg, hauj lwm, daim ntawv
Nyob rau hauv dab tsi daim ntawv no yog manufactured nyob rau hauv kev saib xyuas tshuaj noj? Yuav ua li cas nws hais tias nyob rau cov lus qhia rau kev siv? "Albarel" - ib puag ncig, biconvex ntsiav tshuaj ntawm dawb xim, uas muaj tib lub engraving rau ob sab nyob rau hauv daim ntawv ntawm «H» kos npe rau.
Cov tshuaj yog tau ntim rau hauv cov hlwv ntawm 10 daim thiab ib tug cardboard lub thawv, ntsig txog.
Yuav ua li cas yuav muab "Albarel" tshuaj? Cov lus qhia rau kev siv qhia tias tam sim no lub caij ntawm lub cuab tam yog rilmenidine. Nws kuj muaj xws li tsaug zog accessory cov khoom xyaw li sodium carboxymethyl starch, MCC, khoom paraffin, lactose, magnesium stearate, colloidal anhydrous silica, talc thiab dawb beeswax.
pharmacology
Yuav ua li cas yog raug xa mus rau cov tshuaj? Yuav ua li cas nws hais tias nyob rau cov lus qhia rau kev siv? "Albarel" yog ib qho antihypertensive neeg sawv cev thiab ib tug oxazoline derivative.
Tom qab ua ntawv thov cov tshuaj nkag mus rau hauv kev sib raug zoo nrog imidazoline receptors nyob rau hauv lub peripheral thiab cortical vasomotor chaw zov me nyuam, nrog rau lub raum chaw zov me nyuam. rilmenidine sis raug zoo nrog cov ntsiab txhawb rau inhibition ntawm peripheral sympathomimetic kev ua si thiab cortical chaw zov me nyuam, uas thaum kawg ua rau cov txos ntawm cov ntshav siab.
nta tshuaj
Kev npaj "Albarel" analogs, cov lus qhia rau kev siv uas yog hais hereinafter, nws muaj ib tug hypotensive nyhuv (nyob ntawm seb lub txais txhais tau tias ntawm dosing) rau systolic thiab diastolic ntshav siab nyob rau hauv ib tug sawv los dag txoj hauj lwm. Nws yog muaj pov thawj hais tias thawj coj ntawm cov tshuaj ntawm tshuaj txhaj koob tshuaj (i.e., 1 los yog 2 mg ib hnub twg) yog siv los kho mob loj tsawv rau me me tawg.
Raws li cov kws txawj, cov nyhuv ntawm no neeg sawv cev yog muab thaum lub sij hawm ib hnub. Ntxiv mus, nws yog tshwj xeeb yog zoo thaum lub sij hawm ib ce muaj zog.
Heev siv ntawm cov tshuaj tsis ua yees.
thaj chaw ntawm cov tshuaj
Yuav ua li cas yog zoo tshaj plaws yog cov txhais tau tias raws li "Albarel"? Cov lus qhia rau kev siv, tiag tiag cov kws txawj qhia tias qhov no tshuaj ntawm tshuaj txhaj koob tshuaj tsis cuam tshuam rau hauj lwm ntawm lub plawv, thiab tsis ua rau ncua sij hawm ntawm dej thiab sodium nyob rau hauv lub cev thiab tsis disturb tus metabolic tshuav nyiaj li cas.
Qhov no tshuaj thiaj li peripheral vascular kuj tsis muaj kev hloov nyob rau hauv mob tso zis. Nws yuav tsum tau muab sau tseg tias electrophysiological indexes thiab myocardial contractility nyob rau hauv cov neeg mob uas tau txais cov tshuaj no nyob twj ywm unchanged.
Xam tias yog antihypertensive tshuaj tsis ua orthostatic hypotension (nrog rau cov neeg laus), muaj tsis muaj cov nyhuv rau lub raum ntshav txaus, tsis disturb tus physiological tshua (nyiaj) lub plawv dhia rau ib ce muaj zog, thiab tsis cuam tshuam rau cov roj thiab carbohydrate pauv, pom feem thiab glomerular filtration.
kinetics
Puas "Albarel" tshuaj yog absorbed? Cov lus qhia rau Siv hais tias tus hais tias cov tshuaj no kiag li thiab sai heev absorbed los ntawm cov hnyuv. Tom qab ib tug tib koob tshuaj cai tom qab 2 chasa nws siab tshaj plaws tshuaj concentration nyob rau hauv ntshav.
Lub meej bioavailability ntawm cov tshuaj yog 100%. Nws yuav tsum raug sau tseg hais tias nws yog tsis raug mus rau ua ntej dhau los lub siab.
Cov equilibrium lub xeev ntawm tus neeg mob yog tsim tsuas nrog peb hnub ntawm cov kev kom tsawg ntawm cov ntsiav tshuaj. Cov neeg uas kub siab uas yog nyob rau hauv kev kho mob rau ob peb xyoos, lub concentration ntawm cov tshuaj nyob rau hauv ntshav yog ruaj khov.
Qhov no tshuaj yog tas nyob rau hauv niam cov kua mis. Nws metabolites pom nyob rau hauv cov zis xwb nyob rau hauv txoj lw nyiaj. ib nrab-lub neej ntawm cov tshuaj yuav siv sij hawm txog 8 teev. Qhov no lub sij hawm tsis hloov txawm yog hais tias tus re-lub sij hawm ntawm cov ntsiav tshuaj.
zaj lus tim khawv
Nyob rau hauv tej rooj plaub, cov tshuaj yog tshuaj rau cov neeg mob txog qhov ntawd? Yuav ua li cas nws hais tias nyob rau cov lus qhia rau kev siv? "Albarel" - yog ib tug antihypertensive neeg sawv cev, uas yog muaj kev koom siv nyob rau hauv tawg.
Bans lub sij hawm
Siv yeeb tshuaj "Albarel" yog txwv tsis pub nyob rau hauv:
- cev xeeb tub;
- loj nyuaj siab;
- raum tsis ua hauj lwm (mob loj heev);
- kev pub niam mis;
- Npau taws me ntsis rau rilmenidine los yog lwm yam ntawm cov tshuaj.
Nws yuav tsum tau muab sau tseg tias cov tshuaj no yog tsis siv nyob rau hauv xyuas xyaum.
Ntsiav tshuaj "Albarel": cov lus qhia rau kev siv
Kev kho mob ntawm no lub cuab tam yuav tsum tau pib tsuas yog tom qab kev sib tham nrog tus kws kho mob. Yog hais tias tus neeg mob yog tsis tau mus nrog koj tus kws kho mob ua ntej yuav noj cov tshuaj yuav tsum nyeem cov lus qhia kom zoo zoo. Raws li nws, nyob rau hauv thiaj li yuav ua tau tus yam nyhuv, tus neeg mob txaus noj ib ntsiav tshuaj ua ntej noj tshais. Yog hais tias qhov no ntau npaum "Albarel" tsis txhim kho cov mob ntawm tus neeg mob, ces nws tau nce mus rau 2 ntsiav tshuaj ib hnub twg (coj lub hnub ua ntej noj tshais thiab noj hmo).
xam tau tias yog ib tug txhais tau tias ntawm ntev-lub sij hawm kev kho mob.
Txawm tias muaj tseeb hais tias cov abolition ntawm cov tshuaj no tsis feem ntau ua rau muaj kev phiv, discontinuation ntawm txoj kev kho yuav tsum tau gradual, nrog ib tug gradual yuav txo tau nyob rau hauv koob tshuaj.
Kev nqis tes ua los ntawm-cim
Yuav ua li cas yog cov kev phiv yog suav tias yog antihypertensive neeg sawv cev? Yuav ua li cas hais txog neeg pab leg ntaubntawv qhia rau kev siv? "Albarel" yuav ntxias xws undesirable phenomena li:
- palpitations, orthostatic hypotension, cov nyhuv ntawm no extremities (nyob rau hauv uas tsis tshua muaj neeg mob);
- asthenia, nce qaug zog thaum lub sij hawm ib ce muaj zog, nkees nkees, ntxhov siab vim, insomnia los yog kev nyuaj siab, convulsions (nyob rau hauv uas tsis tshua muaj neeg mob);
- xeev siab, epigastric mob, cem quav, dryness nyob rau hauv lub qhov ncauj, raws plab;
- khaus, daim tawv nqaij ua pob liab vog.
Peb kuj yuav tsum nco ntsoov tias thaum noj cov tshuaj no, ib co neeg mob tej peripheral edema, kub flashes thiab kev sib deev kawg.
overdose txhais tau tias
Yuav ua li cas yuav tshwm sim thaum uas siv cov ib tug loj tus naj npawb ntawm "Albarel" ntsiav tshuaj? Cov lus qhia rau kev siv, koob tshuaj no neeg sawv cev tau hais saum toj no. Yog hais tias koj ntau tshaj qhov tas los tus neeg mob tej zaum yuav tsim kev mob loj hypotension thiab ntau yam kev ua txhaum nyob rau hauv lub psyche. Nyob rau hauv cov ntaub ntawv no, tus neeg muab pais plab lavage thiab nqa sympathomimetic txoj kev kho.
Sis nrog lwm yam tshuaj
Nws tsis pom zoo kom coj "Albarel" tshuaj nrog haus dej haus cawv thiab Mao inhibitors. nram qab no ces xam tau tias yog tshuaj yeeb tshuaj cov kev sib tshuam tau lawm tias raws li cov kws txawj:
- nrog diuretics, antihistamines thiab vasodilators tshwm sim potentiation nyhuv uas cov tshuaj;
- nrog tricyclic antidepressants cim txo antihypertensive nyhuv uas cov tshuaj;
- nrog tshuaj uas inhibit qhov kev txiav txim ntawm lub hauv paus poob siab system, tsaug zog cai.
tej ntaub ntawv
Yog hais tias cov tshuaj no yog siv los ntawm cov neeg uas nyuam qhuav tau muaj ib tug mob stroke los yog heart attack myocardial infarction, rau lawv yuav tsum tau tas li kho mob saib xyuas.
Nyob rau hauv view ntawm lub zoo siab tev taus ntawm lub ntsiav tshuaj 'Albarel "yuav siv tau nyob rau hauv cov neeg mob ntawm advanced muaj hnub nyoog thiab cov neeg mob uas mob ntshav qab zib mellitus.
Yog hais tias koj xav kom txhob muaj cov kev kho mob, cov tshuaj ntau npaum yuav tsum raug txo maj. Nws yuav tsum tau nco ntsoov tias twb nyob rau hauv Feem ntau, lub abolition ntawm cov tshuaj yog tsis tau nrog los ntawm tej yam tshwm sim.
Nws yog txwv tsis pub mus muab "Albarel" ib txhij nrog Mao inhibitors thiab haus dej haus cawv muaj khoom.
Soj ntsuam cov ntaub ntawv rau miv nyuas siv zug thiab kev nyab xeeb ntawm cov tshuaj nyob rau hauv cov me nyuam thiab cov tub ntxhais hluas yog tsis txaus. Nyob rau hauv no hais txog, muab cov tshuaj rau cov neeg mob no yuav tsum tsis txhob yuav.
Thaum kho koob tshuaj "Albarel" muaj tsis ntxim rau psychomotor tshua tib neeg. Yog hais tias cov tshuaj yog kis nyob rau hauv loj tus xov tooj los yog nrog tshuaj, oppressive central lub paj hlwb kev ua si, nyob rau hauv uas cov ntaub ntawv rau tus neeg mob yog txwv tsis pub tsav tsheb tsheb, raws li zoo raws li nyob rau hauv koom lwm yam kev ua ub no.
Analogs thiab xyuas
Analogs tau suav hais tias yog tshuaj yog tsis heev npaum li cas. Ntawm cov feem ntau pheej yig thiab nrov tshaj plaws yog "Tenaksum". Qhov no medicament kuj yog ib qho antihypertensive neeg sawv cev teej tug mus rau cov pab pawg neeg oxazolines. Nws muaj ib tug uas zoo sib xws daim ntawv teev cov contraindications thiab kev phiv, tab sis yog kim kim.
Nrog kev xav txog cov lus ntawm cov neeg mob txog cov tshuaj no, lawv yog ob peb tug. Zoo li cov kws kho mob, tau txais kev pab hais tias nws yog heev txhais tau tias zoo rau tshem tawm tawg. Raws li rau txoj hauj lwm zoo ntawm cov tshuaj muaj xws li nws ntev-lub sij hawm kho nyhuv, xws li thaum lub sij hawm ib ce muaj zog.
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