Noj qab haus huv, Npaj
"Ganaton": li cas ua hauj lwm, yuav ua li cas ua? Xyuas "Ganaton"
Yuav ua li cas yog xws li ib tug yeeb tshuaj raws li "Ganaton"? Nyob rau dab tsi ua rau qhov cuab tam? Cov lus teb rau cov lus nug yuav muaj nyob rau hauv no tsab xov xwm. Koj kuj yuav tau kawm txog dab tsi lub tswv yim yog qhia los ntawm cov neeg mob nyob rau hauv cov tshuaj no, yog hais tias nws muaj tej yam contraindications, thiab yuav ua li cas nws yuav tsum tau coj kom zoo.
Daim ntawv ntawm cov tshuaj, lawv ntim, qauv, hauj lwm
Nyob rau hauv dab tsi daim ntawv no yog manufactured tshuaj "Ganaton"? Cov lus qhia, cov lus sib cav hais tias xws li ib tug tshuaj rau yuav yuav nyob rau hauv daim ntawv ntawm cov ntsiav tshuaj, uas yog dawb, plhaub (zaj duab xis), ib puag ncig puab, cov engraving «HC 803" rau ntawm ib sab thiab txoj kev pheej hmoo - nyob rau lwm yam.
Lub active ingredient ntawm ib tug medicament yog suav tias yog itopride hydrochloride. Raws li koom haum pab constituent yog ib tug yeeb tshuaj muaj xws li lactose, carmellose, pob kws starch, acid, silicic anhydrate, macrogol 6000, magnesium stearate, titanium dioxide, hypromellose, thiab carnauba ciab.
Nyob rau hauv lub qhov muag ntawm xws ntsiav tshuaj tuaj nyob rau hauv sawv hlwv packs, uas nyob rau hauv lem yog fej nyob rau hauv packs ntawm cardboard.
Cov kev khiav hauj lwm hauv paus ntsiab lus ntawm cov tshuaj
Yuav ua li cas yog ib tug "Ganaton"? Nyob rau dab tsi ua rau cov tshuaj no? Nws yog siv los txhim khu hnyuv kom thiab cov laus.
Raws li cov active ingredient ntawm no neeg sawv cev ua itopride hydrochloride. Qhov no tshuaj uas ua rau lub sab sauv txoj kev ntawm lub digestive system, thiab accelerates qhov kev tshem tawm ntawm cov zaub mov ntawm lub plab. Nws yuav tsum tau muab sau tseg tias cov qhia txog kev tivthaiv yog muaj peev xwm muab antiemetic nyhuv.
Lub zog ntawm cov tshuaj
Yuav ua li cas yog zoo tshaj plaws yog cov txhais tau tias raws li "Ganaton"? Nyob rau dab tsi ua rau nws, peb mam li mus ntxiv.
Saib medicament yog ib tug stimulator ntawm kev tso tawm ntawm acetylcholine. Nws lub ntsiab muaj activates pais plab kom (propulsion). Nws tshwm sim vim kev thaiv kev nrog dopamine D2-receptor, thiab koob tshuaj-dependent inhibition ntawm acetylcholinesterase kev ua si.
Itopride hydrochloride activates acetylcholine tso tawm, thiab kuj cheeb nws degradation.
Kev tig tau nta medicament
Nyob qhov twg lub haum ntawm xws li ib tug yeeb tshuaj raws li "Ganaton"? Cov lus qhia rau kev siv, xyuas hais tias cov active ingredient ntawm cov tshuaj sai heev thiab yuav luag tag absorbed los ntawm lub plab. Nws tus kwv tij bioavailability yog kwv yees li 60%. Qhov no yog vim cov tshuaj metabolism, uas tshwm sim nyob rau hauv thawj pass los ntawm lub siab. Khoom noj khoom haus kom tsawg tsis muaj kev ntxim rau cov bioavailability ntawm tus neeg saib xyuas.
Tom qab siv (qhov ncauj) 50 mg itopride hydrochloride concentration ncov yog tiav tom qab 0.5-0.75 sij hawm thiab yog hais txog 0,28 ug / ml. Ua kom tsawg ntawm cov tshuaj rau ib koob tshuaj 50-200 mg peb zaug ib hnub twg rau ib lub lim tiam yog linear tshuaj. Nyob rau hauv cov ntaub ntawv no, cia hnab khib yog tsawg heev.
Kev sib txuas lus tshuaj rau ntshav cov nqaijrog yog kwv yees li 96%. Nws yog kev koom faib nyob rau hauv tag nrho cov ntaub so ntswg thiab yog pom nyob rau hauv siab ntau nyob rau hauv lub siab, mob raum, adrenal caj pas, hnyuv, thiab lub plab. Tshuaj penetrates cov ntshav-hlwb barrier nyob rau hauv me me nyiaj. Nws kuj stands nrog leej niam cov kua mis.
Feem itopride hydrochloride thiab nws cov derivatives muaj tshwm sim nrog cov zis. Raum feem ntawm lub active tshuaj tom qab tau txais ib tug tib kho koob tshuaj yog hais txog 75%. Qhov kawg ib nrab-lub neej ntawm no neeg sawv cev yog hais txog rau lub sij hawm.
Tshuaj "Ganaton": dab tsi pab?
Qhov cuab yeej no yog dav siv nyob rau hauv cov kev kho mob ntawm gastro-plab hnyuv teeb meem uas yog txuam nrog uas tsis yog-rwj haumxeeb dyspepsia (xws li mob gastritis), raws li zoo raws li ncua pais plab kom.
Yog li ntawd thaum twg siv cov tshuaj "Ganaton"? Daim ntawv thov ntawm no txhais tau tias yog qhia nyob:
- anorexia;
- tsam plab;
- kub siab;
- ntuav;
- lawm ntawm fullness nyob rau hauv lub plab tom qab ib tug noj mov;
- mob los yog tsis xis nyob rau hauv lub epigastric cheeb tsam;
- xeev siab.
Txwv tau txais tshuaj
Tam sim no, koj paub, dab tsi yog zoo tshaj plaws yog cov txhais tau tias raws li "Ganaton". Los ntawm tej yam, khoom kev npaj no, peb kuj pom. Nws yuav tsum tau qhia tias cov kev kawm tshuaj no yog txhob tau txais nyob rau hauv:
- cev xeeb tub;
- hnyuv los ntshav, neeg kho tshuab rhuav txhua los yog perforation ntawm tus mob huam;
- nyob rau hauv lub hnub nyoog ntawm 16 xyoo;
- kev pub niam mis;
- npau taws me ntsis rau Itopride los yog lwm yam koom haum pab tshuaj.
Ceev faj npaj txais tos
Lub cuab tam tshuaj nrog ceev faj cov neeg laus vim hais tias ntawm lub heev yuav txo tau nyob rau hauv ob lub raum thiab lub siab, raws li tau zoo raws li concomitant kab mob los yog lwm yam kev kho mob.
Tshuav rau potentiation ntawm acetylcholine medicament xam tau tias yog nrog ceev faj kom koj hais tias cov neeg mob uas tsim cholinergic tshwm sim muaj paug thaum lub sij hawm lub ntsiab kab mob.
Yuav ua li cas tau "Ganaton"?
Xam tias yog ntsiav tshuaj yuav tsum tau coj lus ua ntej noj mov. Lawv ntxuav cia nrog dej dawb.
Cov tshuaj muaj tsis muaj cov nyhuv rau ib tug neeg muaj peev xwm tsav tsheb, raws li zoo raws li txoj mechanisms. Thaum uas siv cov "Ganaton" neeg laus los yog cov neeg uas muaj kev zoo raum muaj nuj nqi thiab siab lawv yuav tsum tau tas li kho mob saib xyuas.
Tej zaum tus kws kho mob tej zaum yuav nqa tawm kho ntawm lub pom zoo npaum li cas. Yog hais tias ntawd nqos ib tug loj npaum li cas ntawm cov tshuaj yuav tsum tau rau kev xws txheem kev ntsuas raws li symptomatic kev kho mob, thiab pais plab lavage.
Nyob rau hauv dab tsi ntau npaum tus neeg mob yuav tsum tau noj cov tshuaj "Ganaton"? Daim ntawv thov (xyuas ntawm cov tshuaj yuav sib tham txog hauv qab no) no txhais tau tias koj yuav tsum tau nqa tawm tom qab kev sib tham nrog tus kws kho mob. Lub sij hawm ntau npaum ntawm cov tshuaj nyob rau hauv kev saib xyuas rau cov neeg laus yog 150 mg. Yog hais tias tsim nyog, lub saum toj no ntau npaum li cas tej zaum yuav hloov los ntawm ib tug neeg txawj.
Raws li ib tug txoj cai, qhov cuab tam yog pom zoo kom noj peb zaug ib hnub twg, ib tug ntsiav tshuaj ua ntej noj mov (50 mg). Lub caij ntawm kev kho mob yog txiav txim los ntawm tus kws kho mob thiab tej zaum yuav txog 5-8 lub lis piam.
txiav txim sab
Yuav ua li cas cov tshuaj tiv thaiv los ntawm qhov yuav ua rau cov tshuaj "Ganaton"? Qhov no yuav pab tshuaj plurality hnyuv kab mob, tab sis tej zaum nws yuav ntxias cov nram qab no undesirable los:
- Endocrine System: gynecomastia, nce prolactin theem.
- hemopoietic system: thrombocytopenia, leukopenia.
- Cov kev tsis haum: daim tawv nqaij khaus, lossis puas liab liab ntawm daim tawv nqaij, anaphylaxis, tawm pob.
- Cns: mob taub hau, kiv taub hau, co.
- Hnyuv: daj ntseg, raws plab, muaj zog qaub ncaug, cem quav, xeev siab, mob plab.
- Cov kev hloov nyob rau hauv laboratory tsom xam: nce theem ntawm bilirubin thiab alkaline phosphatase, raws li zoo raws li cov kev ua ntawm ALT, AST thiab GGT.
tshuaj cov kev sib tshuam
Metabolic kev sib tshuam ntawm cov tshuaj no yog tsis tau. Qhov no yog vim lub fact tias itopride metabolized tsis tus isozymes ntawm cytochrome P450, thiab nyob rau hauv qhov kev txiav txim ntawm flavin monooxygenase.
Lub active tshuaj yog suav hais tias yog tshuaj tsub kom lub kom ntawm lub plab, uas muaj peev xwm muaj kev cuam tshuam cov haum lwm qhov ncauj tshuaj siv ib txhij. Ceev faj yuav tsum tau coj thaum noj tshuaj nrog ib tug tsawg kho index. Tib yam siv rau kev npaj nrog enteric coated pab tawm formulations thiab lub ntsiab tivthaiv.
Thaum combining "Ganaton" nrog "Diazepam", "warfarin", ticlopidine hydrochloride, diclofenac sodium, nicardipine hydrochloride thiab "nifedipine" itopride hloov nyob rau hauv lub ruaj rau ntshav cov nqaijrog muaj cai.
Anti-rwj tshuaj xws li "Ranitidine", "cimetidine", "cetraxate" thiab "teprenone" tsis cuam tshuam rau kinetics ntawm lub Itopride.
Anticholinergic tshuaj tsis muaj zog cov nyhuv uas cov active tshuaj nyob rau hauv kev saib xyuas txhais tau tias.
Khoom noj khoom haus thiab cev xeeb tub
Tam sim no, tsis txaus cov ntaub ntawv hais txog kev siv ntawm Itopride hydrochloride thaum lub sij hawm cev xeeb tub tsis tau. Kev siv cov no lub cuab tam nyob rau hauv tus txheej txheem ntawm hnub no tsuas tau nyob rau hauv lub qhaj ntawv ntawm lwm txoj kev kho mob, raws li tau zoo raws li lub peev xwm pab rau tus niam, uas yog ntau tshaj qhov uas yuav kom cov me nyuam hauv plab.
Nws yuav tsum tau muab sau tseg tias thaum lub sij hawm kev kho mob nrog cov tshuaj no muaj ib tug uas yuav mob tshwm sim nyob rau hauv tus me nyuam mos. Nyob rau hauv no hais txog, qhov yuav tsum tau siv cov tshuaj nyob rau hauv lub mis-pub lub sij hawm ntawm lactation yuav tsum tau txiav.
Zoo li txhais tau tias thiab cov tshuaj nqi
Yog koj paub ntau npaum li cas nws cov nqi ua ntej peb tshuaj? Yog hais tias tej ntaub ntawv koj tsis muaj, peb yuav muab rau koj. Tus nqi ntawm qhov cuab tam nyob rau hauv lub paj tau paj, thiab cov thawj-aid network yog hais txog 250 rubles rau 10 ntsiav tshuaj.
Yog hais tias cov tshuaj tsis pom nrog tib lub npe, nws puas yuav tau los hloov analogue. Cov xws tshuaj yog cov tshuaj mas siv nrog cov tib yam kom nquag plias yam khoom uas, uas yog, nrog Itopride. Raws li lawv feem ntau siv "Itomed", "Itopride", "Itopru" thiab "Primer".
Xyuas ntawm cov neeg mob thiab cov tub txawg
Puas "Ganaton" nrog Helicobacter pylori? Kws txawj qhia tias deals nrog cov txhais tau tias yog ib cov tshuaj uas pab txoj kev lub suab nrov thiab kom ntawm lub digestive ib ntsuj av. Qhov no tsis yog ib qho antibacterial tshuaj uas muaj peev xwm kov yeej lub saum toj no-hais kab mob. Txawm li cas los, nyob rau hauv tej zaum nws yog tseem muab nyob rau hauv tus kab mob no, tab sis tsuas nyob rau hauv ua ke nrog txoj kev kho nyob rau hauv nrog tshuaj tua kab mob thiab lwm yam anti-rwj ceev dua.
Yuav luag tag nrho cov neeg uas tau puas tau xam tau tias yog kev noj tshuaj, tham txog nws cov high efficiency. Raws li lawv, tom qab traversed ib chav kawm ntawm txoj kev kho ntawm cov tshuaj eliminates cov kev xav ntawm xeev siab thiab tsis xis nyob nyob rau hauv lub epigastric cheeb tsam, raws li zoo raws li qhov nyhav thiab mob nyob rau hauv lub plab.
Ib txhia neeg teb zoo rau qhov no medicament raws li ib tug kev npaj rau cov tshem tawm ntawm episodic kub siab thiab ntuav.
Nrog hais txog lus ceeb toom ntawm kev phiv tshuaj "Ganaton", lawv tsis tshua muaj. Raws li ib tug txoj cai, nyob rau hauv cov neeg mob uas tau txais no neeg sawv cev nyob rau hauv ib co neeg mob muaj yog nce salivation, nkees nkees los yog kiv kiv taub hau.
Xyuas ntawm overdose mob no lub cuab tam tsis tau tas kom deb li deb. Tus nqi ntawm xws formulation li "Ganaton" ntaus nqi los ntawm kev pab raws li ib tug tau los yog siab.
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