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Cov tshuaj "Efferalgan" (taws tswm ciab) - zoo analgesic thiab antipyretic
"Efferalgan" (taws tswm ciab) sawv cev rau cov tshuaj uas muaj analgesic thiab antipyretic nyhuv. Lub active compound nyob rau hauv hais tias formulation yog paracetamol, uas koom rau uas tsis yog-tshuaj cov neeg ua hauj. Tshuaj "Efferalgan 150" niamntiav nws cov nyhuv los ntawm qhov tseeb hais tias muaj yog tsis yog-xim inhibition ntawm cyclooxygenase enzyme ua si yog li ntawd txo cov synthesis ntawm prostaglandins los ntawm arachidonic acid. Txij li thaum lub txo tus naj npawb ntawm prostaglandins, muaj yog ib tug txo nyob rau hauv lub central lub paj hlwb mob impulses. Ib tug antipyretic nyhuv, uas muaj "Efferalgan" -svechi yog tiav vim lub fact tias paracetamol muaj feem xyuam rau thermoregulation chaw nyob rau hauv lub hypothalamus.
Qhov no tshuaj yog ua nyob rau hauv daim ntawv ntawm cov ntsiav tshuaj thiab syrups, los yog nyob rau hauv daim ntawv ntawm cov suppositories. Nws sai sai absorbed ntawm lub cev thiab nws cov nyhuv twb 20 feeb tom qab nkag mus rau hauv lub cev. Qhov siab tshaj plaws concentration ntawm paracetamol nyob rau hauv cov ntshav yog mus txog tom qab 30-55 feeb tom qab nws tau tau ua tswvcuab "Efferalgan" -svechi. Cov tshuaj no yog metabolized nyob rau hauv lub siab, lub pharmacologically tsaug zog metabolites raug tsim. Tas metabolites muab siv rau ob lub raum. Qhov nruab nrab ib nrab-lub neej ntawm cov tshuaj "Efferalgan" (taws tswm ciab 150 mg) los ntawm lub cev tshwm sim los ntawm 2 teev thiab ib hnub twg tom qab twb tso tawm mus txog 90% ntawm cov khoom paracetamol.
Pom zoo rau kev siv cov tshuaj "Efferalgan"
Taws tswm ciab yog siv rau cov kev kho mob ntawm cov me nyuam muaj hnub nyoog 3-5 lub hlis, uas 6 kilograms nyob rau hauv cov nram no mob:
- nyob rau hauv lub xub ntiag ntawm ib tug me nyuam lub siab kub, uas yog tshwm sim los ntawm ua pa kab mob, kab mob khaub thuas, los yog lwm yam kab mob thiab cov kab mob inflammatory;
- raws li ib tug ua kom loog, yog tias muaj mob los yog mob me me mus tsawv siv, nws yuav tshwm sim thaum poob plig mob, mob ib ce, kub nyhiab, lub taub hau thiab mob hniav, neuralgia.
Cov tshuaj "Efferalgan" (taws tswm ciab) - txoj kev ntawm daim ntawv thov thiab pom zoo ntau npaum
Taws tswm ciab yog muab rectally. Ua li no, tau ib tug tswm ciab los ntawm nws cov ntim thiab ua tib zoo qhia koj tus me nyuam lub qhov quav, ua ntej nws yuav tsum tau ua los yog enema, los yog tos rau txawj plob tsis so tswj zog.
Ib tug tib koob tshuaj hais tias formulation nyob rau tus me nyuam thiab tus luj yuav tsum 10-15 mg / kg, xeem "Efferalgan" -svechi 3 mus rau 4 lub sij hawm ib hnub. Thoob plaws hauv lub hnub koj yuav tsis tau ntau tshaj li 60 mg / kg ntawm cov tshuaj.
Rau cov me nyuam hnub nyoog 3-5 lub hlis, nws yog tsim nyog los siv 1 suppository (80 mg), los ntawm 6 lub hlis mus rau 3 xyoos - 1 suppository 150 mg, los ntawm 5 mus rau 10 xyoo - 1 suppository 300 mg ntawm cov tshuaj. Lub caij nyoog nruab nrab tshuaj yuav tsum nyob nruab nrab ntawm 4 thiab 6 teev.
Feem ntau, kev kho mob yog txuas ntxiv mus rau 3 hnub yog hais tias tus yeeb tshuaj yog siv los txo qhov kub thiab mus txog rau 5 hnub, yog hais tias nws yog siv raws li ib tug ua kom loog. Yog hais tias koj yuav tau siv cov tshuaj rau ib tug ntev lub sij hawm, nws yog tsim nyog los soj ntsuam daim siab muaj nuj nqi thiab saib xyuas tus txheej xwm ntawm peripheral cov ntshav.
Tsis tas li ntawd lub cuab tam yuav siv tau nyob rau hauv daim ntawv ntawm ib tug phoov los yog soluble cov ntsiav tshuaj. Lub caij ntawm kev kho mob kho los ntawm ib tus kws kho mob, tiam sis nws yuav tsum tau xyuas kom muaj hais tias cov hnub koob tshuaj paracetamol yuav tsum tsis txhob ntau tshaj cov muaj hnub nyoog txwv (tsis hais txog ntawm daim ntawv nyob rau hauv uas nws yog noj).
Tau tshwm sim los ntawm cov tshuaj "Efferalgan"
Feem ntau cov teeb meem tom qab tau txais no formulation tsis tshwm sim. Nyob rau hauv tsawg tus neeg mob, tej zaum yuav ua rau xeev siab thiab ntuav, thiab hypotension, allergic daim tawv nqaij tshua, qaug zog thiab kiv taub hau.
Contraindications
Tsis txhob noj cov tshuaj no txhais tau hais tias cov neeg uas muaj mob loj heev siab los yog raum kab mob, raws li tau zoo raws li cov neeg uas tsis tau tso fructose thiab quav dej quav cawv. Yog hais tias tus me nyuam yog yau dua 2 xyoos uas muaj hnub nyoog los yog tsis nyhav tshaj 13 kilograms, lub effervescent ntsiav tshuaj kuj tsis pom zoo. Cov tshuaj "Efferalgan" (taws tswm ciab) yog tsis siv nyob rau hauv cov neeg mob uas muaj tsis ntev los raug kev txom nyem mob (los yog los ntshav) ntawm lub qhov quav. Nyob rau hauv cov ntaub ntawv no, zoo dua yuav xaiv lwm daim ntawv ntawm cov tshuaj.
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