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Analogue "Diflucan" - txhais tau tias "Fluconazole"

Analogue "Diflucan" - txhais tau tias "Fluconazole" - yog ib tug noj neeg sawv cev muaj ib tug heev cov kev nyhuv. Cov tshuaj uas muaj peev xwm ntawm thaiv cov hlab cov kev ua ntawm ib co enzymes, inhibit transformation ntawm lanosterol rau ergosterol. Nyob rau hauv tas li ntawd, cov tshuaj yuav tsub kom lub permeability ntawm cell week, tiv thaiv replication thiab kev loj hlob ntawm pathogens. Cov tshuaj no yuav siv tau rau opportunistic fungal kab mob provoked los ntawm fungi genus Candida, xws li generalized tiv thaiv hom Candidiasis nyob rau hauv cov av. Nrog qhov ncauj tshuaj muaj zoo absorbability. Thaum tus nqi ntawm haum yog tsis cuam tshuam los ntawm khoom noj khoom haus kom tsawg. Lub bioavailability ntawm cov tshuaj yog hais txog 90%. Maximum cov ntsiab lus nyob rau hauv cov ntshav nce mus txog ib tug kho nyob rau hauv 30-90 feeb. Cov tshuaj no yog zoo faib nyob rau hauv cov ntaub so ntswg thiab kua txeem mus rau hauv cov mis nyuj. Nws yuav tsum tau hais tias tus nqi ntawm cov tshuaj "Fluconazole" qho kev txiav txim ntawm qhov ntau tsawg dua tus nqi ntawm "Diflucan" (nyob rau hauv lub yav dhau los yuav tau them los ntawm plaub puas yim puas rubles).

zaj lus tim khawv

Tshuaj "Fluconazole" (analogue "Diflucan") yog muab nyob rau hauv cryptococcal meningitis, cryptococcosis thiab lwm yam localizations cryptococcal kab mob nyob rau hauv cov neeg mob uas muaj ib tug ib txwm tiv thaiv kab mob teb thiab nrog ntau hom tiv thaiv. Los ntawm cov lus tim khawv ntawm Candidiasis xws li generalized hom, disseminated Candidiasis, candidemia, thiab lwm yam kev tus kab mob tshwm sim los ntawm ib cov pwm Candida. Cov tshuaj yog pom zoo rau cov kev tiv thaiv ntawm fungal kab mob nyob rau hauv cov neeg mob uas phem hlav ntawm cov ua cim. Yam uas luag muab neeg sawv cev rau mycosis taw, puab tais, npog tas ib ce.

dosing regimen

Analogue "Diflucan" - txhais tau tias "Fluconazole" - tshuaj rau cov neeg mob nrog kaum tsib xyoos nyob ib tug loj ntau dua li 50 kg. Thaum cryptococcal kab mob sib txawv ntawm cov localization nyob rau hauv thawj hnub ntawm ib koob tshuaj ntawm 400 mg. Tom qab, tus nqi ntawm cov medicament txo rau 200 mg ib hnub twg. Duration ntawm kev kho nyob rau hauv cov pathologies nyob rau hauv lub efficiency ntawm cov kev kho mob, uas yog paub tseeb hais tias los ntawm mycological kev tshawb fawb. Daim ntawv thov ntawm cryptococcal meningitis yuav tsum kav tsawg kawg yog rau mus rau yim lub lim piam. Thaum disseminated Candidiasis, candidemia, thiab lwm yam kev tus Candida kab mob nyob rau hauv thawj hnub tus nqi ntawm cov tshuaj - 400 mg, ntau npaum yuav txo rau 200 mg. Nyob rau hauv cov ntaub ntawv ntawm txaus los khi cov hauj lwm zoo ntawm kev kho mob ntau npaum yog nce rov qab mus rau 400 mg. Lub caij ntawm kev kho mob nyob rau cov hauj lwm zoo ntawm cov txhais tau tias.

sab nyhuv

Analogue "Diflucan" - cov tshuaj "Fluconazole" - yuav ua rau kiv taub hau, mob nyob rau hauv lub taub hau, plab, mob plab, tsis qab los, xeev siab. Nyob rau lub hauv paus ntawm kev kho mob tej zaum yuav tsim thrombocytopenia, allergic kev tig cev xws li o ntawm lub ntsej muag, epidermal lom necrolysis, daim tawv nqaij khaus. Analogs ntsiav tshuaj yuav ua rau muaj kev cuam tshuam ntawm lub siab, raum, hypokalemia, hypertriglyceridemia.

Contraindications

Tsis txhob muab cov tshuaj ua ntej lub hnub nyoog 4 xyoo, nyob rau hauv cov ntaub ntawv ntawm intolerance ntawm nws cov Cheebtsam. Txhob ua ke siv nrog cov medicament "Terfenadine", "Astemizole" thiab lwm yam pab rau lengthening ntawm QT-luv. Ceev faj thaum lub sij hawm txoj kev kho nrog yeeb predisposition mus txawv pathologies (rau ntsha tsis txaus, organic kab mob plawv, thiab lwm yam).

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