Noj qab haus huvNpaj

"Antabuse" tshuaj. Xyuas, nqe phau ntawv

Nws hu ua alcoholism ib tug kab mob uas yog yus muaj los ntawm ib tug tiv rau Ethanol nrog lub cev, thiab puas hawv dependence rau nws. Qhov no zoo ntawm kev tsim txom. Nyob rau hauv lub xeev no, tsis tswj tus nqi qaug dej qaug cawv cawv tsub kom kam rau nws (mus cuag siab cawv lossi ua koob) thiab ntsoos ntsoos syndrome tshwm sim, muaj feem xyuam rau hauv nruab nrog cev thiab tshwm sim nco xyaum.

Cov neeg mob kev txom nyem los ntawm alcoholism, hu ua quav dej quav cawv. Kho tus kab mob no yuav tsum hlwb thiab lub cev. Heev feem ntau, cov kws kho mob muab cov tshuaj no rau cov neeg "Antabuse". Cov lus qhia rau kev siv, tus nqi ntawm cov tshuaj, kev kho mob xyuas yog qhia hauv qab no.

Cov, zoo lawm, thiab cov qauv piav qhia

Nyob rau hauv dab tsi tsim cov tshuaj yog muag "Antabuse"? Testimonials qhia hais tias xws li ib tug tshuaj rau yuav yuav nyob rau hauv daim ntawv ntawm cov dawb, puag ncig effervescent ntsiav tshuaj. Lawv yog ca, beveled ntug, uas yuav muaj thiab cim «CD» thiab «C» rau ob tog ntawm cov kev txaus ntshai.

Muaj pes tsawg leeg ntawm cov tshuaj no muaj xws li disulfiram. Dhau li nws, cov kev npaj muaj pob kws starch, povidone, sodium hydrogencarbonate, tartaric acid, colloidal silicon dioxide, talc, microcrystalline cellulose thiab magnesium stearate.

Ntsiav tshuaj "Antabuse" muab tso rau hauv hnab yas ntim thiab packs cardboard.

pharmacodynamic yam ntxwv

Yuav ua li cas yog cov tshuaj "Antabuse"? Phau ntawv lub xeev hais tias qhov no txhais tau tias antialcoholic. Nws cheeb acetaldehyde dehydrogenase, uas yog muab kev koom tes nyob rau hauv lub metabolism ntawm ethanol. Ncua nws oxidation txheej txheem ua rau lub hnab khib cawv thiab txoj kev loj hlob muaj zog intoxication, ua raws li los ntawm hnyav txoj kev xav raws li ib tug throbbing mob thiab cov suab nrov nyob rau hauv lub taub hau, tachycardia, palpitation, yuav txo tau nyob rau hauv cov ntshav siab, xeev siab, qhov muag plooj tsis pom kev thiab ntuav.

Raws li kws txawj, cov tsis kaj siab tsos mob pab mus rau txoj kev loj hlob ntawm conditioned reflex aversion rau dej cawv.

pharmacokinetic zog

Yuav ua li cas puas muaj tus haum ntawm "Antabuse" tshuaj? Phau ntawv qhia tias cov tshuaj yog absorbed los ntawm 70-80%. Nws yog ib co soluble nyob rau hauv lipids thiab nyhav ntxiv nyob rau hauv cov roj depot.

Lub active tshuaj ntawm tus neeg saib xyuas yog sai heev metabolized, ua nyob rau hauv lub hloov metabolite - methyl ester dietiltiokarbaminovoy acid. Nws ncov ntshav ntau txiav txim tom qab 4 h. Txawm hais tias kev ua si nyob rau hauv relation mus acetaldehyde dehydrogenase yog cai tsuas yog tom qab peb hnub.

Lub ib nrab-lub neej ntawm cov tshuaj yog 10 xuab moos. Ntxiv mus, txoj kev tiv thaiv aldehyde dehydrogenase tsawv ntev npaum li cas. Yog li ntawd, tom qab qhov kev tshem tawm ntawm cov nyhuv uas cov ntsiav tshuaj muaj cai rau ib tug ntxiv 7-14 hnub.

Cov tshuaj zoo nkaus li nyob rau hauv cov zis, thiab tej los ntawm cov hnyuv nrog exhaled cua.

zaj lus tim khawv

Nyob rau hauv tej rooj plaub, qhov zoo tshaj tshuaj behaves "Antabuse"? Xyuas tau tshaj tawm hais tias lub tsev no yog dav siv rau kev tiv thaiv ntawm relapse nyob rau hauv cov kev kho mob ntawm cov cawv dependence thiab alcoholism.

Contraindications

Thaum koj yuav tsum tsis txhob coj "Antabuse" ntsiav tshuaj? Guest cov kws txawj hais tias pom tau hais tias cov tshuaj yuav tsum tsis txhob muab yog hais tias:

  • glaucoma;
  • neuritis ntawm lub optic thiab hnov paj;
  • pulmonary tuberculosis;
  • lub plawv thiab leeg tshav kab mob (e.g., post-infarction lub xeev, qhia cardiosclerosis, atherosclerosis ntawm cerebral hlab ntsha, hypertensive tus kab mob, aortic aneurysm);
  • polyneuritis ntawm tej keeb kwm;
  • mob ntshav qab zib;
  • mob hawb pob, bronchial hawb pob;
  • thyrotoxicosis;
  • kev puas hlwb, qaug dab peg thiab epileptiform syndrome;
  • kab mob qog hlav;
  • mob loj heev hepatic thiab lub raum tsis ua hauj lwm;
  • cov kab mob ntawm hematopoiesis;
  • exacerbation ntawm peptic rwj kab mob;
  • cev xeeb tub;
  • npau taws me ntsis.

Tsis tas li ntawd nco ntsoov hais tias qhov no tshuaj yog txheeb ze contraindications:

  • muaj hnub nyoog ntawm 60 xyoo;
  • cov teebmeem ntawm ib stroke nrog residual cov tsos mob;
  • peptic rwj (xws li nyob rau hauv txoj kev zam txim);
  • precipitates ib psychosis.

Tshuaj "Antabuse": cov lus qhia rau kev siv

Anti-cawv ntsiav tshuaj nqi uas teev tseg nyob rau hauv lub kawg ntawm tsab xov xwm. Yuav tsum coj lawv cov inward ½ yav tas yaj nyob rau hauv ib khob ntawm cov dej.

Feem ntau, cov kws kho mob muab tshuaj rau 200-500 mg ntawm yeeb tshuaj ib zaug los yog ob zaug ib hnub twg. Tom qab 7 hnub, nco ntsoov siv disulfiram-cawv xeem. Nyob rau hauv thaum uas tig mus nrog tus txais tos ntawm 500 mg ntawm medicament neeg mob cov dej qab zib 20-30 ml ntawm vodka. Yog hais tias qhov tshuaj tiv thaiv yog tsis muaj zog, ces kom cov tshuaj cawv mus rau 20 ml.

Qhov no kuaj yog rov qab ob peb lub sij hawm. Tom qab ntawd ballroom tshuaj txij nkawm ntau npaum ntawm 200 mg txhua hnub rau 1-3 xyoos.

phiv tshua

Ntsiav tshuaj "Antabuse", uas kev uas hais hauv qab no tej zaum yuav ua rau cov nram qab no tshwm sim tsis zoo:

  • kab mob siab, asthenia, hlau saj nyob rau hauv lub qhov ncauj;
  • cutaneous ces, polyneuritis ko taw;
  • nco tsis tau, lub hlwb o, mob taub hau;
  • myocardial infarction, mob arrhythmias;
  • ua pa tsis ua hauj lwm, mob plawv cev qhuav dej;
  • optic neuritis, cerebral thrombosis hlab ntsha;
  • psychoses, angina.

Medicament "Antabuse": xyuas ntawm cov kws kho mob thiab cov nqi

Tus nqi ntawm cov anti-cawv ntsiav tshuaj yog hais txog 450-600 rubles (nyob ntawm seb cov tshuaj thiab cov nyiaj ib pob).

Cov kws kho mob uas muab cov tshuaj xws li ib tug yeeb tshuaj, tam sim ntawd ceeb toom ntawm lub loj teeb meem uas yuav tshwm sim nyob rau hauv ib tug neeg mob nyob rau hauv lub keeb kwm yav dhau nws yuav siv sij hawm. Yog li ntawd txwv tsis pub los kho koj tus kheej los yog ib tug tsis pub leejtwg paub los ntawm tus neeg mob.

Nws yuav tsum tau muab sau tseg tias feem ntau cov kws txawj pom zoo hais tias siv tau cov tshuaj uas suppress lub yees rau cawv, tsis muaj. Thiab cov qauv no yog tsis kho. Nws pawg txhawb ib tug ruaj khov kev so ib pliag.

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